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| Protein Kinase Information : List of Protein Kinase Inhibitor | |||||||||||
| # | Name of Kinase | Name of Inhibitor | |||||||||
| 1 | PKA | H-89, HA-1004, H-7, H-8, HA-100, staurosporine | |||||||||
| 2 | PKG | H-7, H-8, HA-1004, H-89 | |||||||||
| 3 | PKC | bisindolylmaleimide IX, chelerythrine, edelfosine, edelfosina, ET18OCH3, H-7, HA-100, H89, HA-1004, Ro 31-8220, staurosporine | |||||||||
| 4 | ABL | PP1 | |||||||||
| 5 | Adenosine kinase | 5-Iodotubercidin | |||||||||
| 6 | Akt/PKB | Triciribine (TCN, Tricyclic Nucleoside, NSC-154020, API-2) | |||||||||
| 7 | AMPK | indirubin-3'-oxime, 5-Iodotubercidin, H-89 | |||||||||
| 8 | BTK | LFM-A13 | |||||||||
| 9 | CaMKII | KN-62, W-7, HA-1004, HA-1077 | |||||||||
| 10 | CDK1, CDK2, CDK5 | aloisine, aloisine A, alsterpaullone, indirubin-3'-oxime, kenpaullone, olomoucine, purvalanol A, roscovitine | |||||||||
| 11 | CHK1 | H-89 | |||||||||
| 12 | CK1 | DRB | |||||||||
| 13 | CK2 | TBB, DRB | |||||||||
| 14 | EGF-R kinase | erbstatin analog, erlotinib, gefitinib, PD 153035, Tyrphostin AG 490, Tyrphostin AG 825, PP1, PP2 | |||||||||
| 15 | ERK kinase | PD 98059, SL327, olomoucine, 5-Iodotubercidin | |||||||||
| 16 | FYN | PP1, PP2, SU6656 | |||||||||
| 17 | GSK3 | aloisine, aloisine A, indirubin-3'-oxime, kenpaullone | |||||||||
| 18 | HCK | PP2 | |||||||||
| 19 | HER2 | Tyrphostin AG 825 | |||||||||
| 20 | IGF1-R PTK inhibitor | Tyrphostin AG 1024 | |||||||||
| 21 | JAK | Tyrphostin AG 490 | |||||||||
| 22 | JNK | aloisine A, SP600125 | |||||||||
| 23 | KIT | PP1 | |||||||||
| 24 | LCK | aminogenistein, PP1, PP2, indirubin-3'-oxime, kenpaullone | |||||||||
| 25 | LYN | SU6656 | |||||||||
| 26 | MAPKAP-K1b | HA-1077 | |||||||||
| 27 | MAPK | SB202190, SB203580 | |||||||||
| 28 | MAPKK | arctigenin, PD 98059, SL327, U0126 | |||||||||
| 29 | MEK | PD 98059, SL327, U0126 | |||||||||
| 30 | MKK | arctigenin, PD 98059, SL327, U0126 | |||||||||
| 31 | MLCK | ML-9, W-7, HA-100, HA-1004, H-7, H-8, HA-1077 | |||||||||
| 32 | MSK1 | H-89, ML-9, HA-1077 | |||||||||
| 33 | P38 MAPK | SB202190, SB203580 | |||||||||
| 34 | PDGF-R kinase | DMPQ | |||||||||
| 35 | PI3K | LY294002 | |||||||||
| 36 | PRK2 | HA-1077 | |||||||||
| 37 | RHO kinase | HA-1077 | |||||||||
| 38 | ROCK | Y-27632, H-89, ML-9, HA-1077 | |||||||||
| 39 | S6K1 | rapamycin, sirolimus, H-89, ML-9, HA-1077 | |||||||||
| 40 | SAPK | PD 169316, SB202190, SB203580 | |||||||||
| 41 | SGK | indirubin-3'-oxime, H-89 | |||||||||
| 42 | SRC familiy PTK | PP1, PP2, SU6656 | |||||||||
| 43 | SYK | piceatannol | |||||||||
| 44 | TOR | rapamycin, sirolimus | |||||||||
| 45 | PTK | aminogenistein, DMPQ, erbstatin analog, erlotinib, gefitinib, LFM-A13, PD 153035, piceatannol, PP1, PP2, SU 4312, SU6656, Tyrphostin AG 490, Tyrphostin AG 825 | |||||||||
| 46 | VEGF-R kinase | SU 4312 | |||||||||
| 47 | YES | SU6656 | |||||||||
| 48 | ZAP70 | piceatannol | |||||||||